Losartan

Losartan

SCHEMBL4677535

CCCCc1nc(Cl)c(CO)n1Cc1ccc(-c2ccccc2-c2nn[nH]n2)cc1.[KH]

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.84
AGTR2 P50052 1/20 0.75
GP6 Q9HCN6 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Losartan SCHEMBL4222 0.99 AGTR1 (0.86) AGTR1AGTR2GP6
SCHEMBL20257387 0.93 AGTR1 (0.81) AGTR1AGTR2GP6
Losartan SCHEMBL14169312 0.92 AGTR1 (0.80) AGTR1AGTR2GP6
Losartan SCHEMBL2577425 0.92 AGTR1 (0.74) AGTR1AGTR2GP6
Losartan SCHEMBL31663637 0.91 AGTR1 (0.73) AGTR1AGTR2GP6
SCHEMBL3633085 0.91 AGTR1 (0.78) AGTR1AGTR2GP6
SCHEMBL8468357 0.89 AGTR1 (0.76) AGTR1AGTR2GP6
SCHEMBL20257373 0.89 AGTR1 (0.76) AGTR1AGTR2GP6
SCHEMBL2615537 0.88 AGTR1 (0.69) AGTR1AGTR2GP6
SCHEMBL2834891 0.88 GP6 (0.77) AGTR1AGTR2GP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527879-B1 SYNERGISTIC THERAPEUTIC COMPOSITIONS AND METHODS PFIZER (US) 1997-02-05 EP claimed
CN-101237892-A Method for conjugating molecules containing an aminothiol to a carrier AMGEN INC (US) 2008-08-06 CN disclosed
EP-1544198-B1 A process for the preparation of crystalline losartan potassium DIPHARMA SPA (IT) 2008-06-04 EP disclosed
EP-1544198-A1 A process for the preparation of crystalline losartan potassium Dipharma S.p.A. (IT) 2005-06-22 EP disclosed
US-20050131040-A1 Process for the preparation of crystalline losartan potassium DIPHARMA S.P.A. (IT) 2005-06-16 US disclosed
EP-0527879-B1 SYNERGISTIC THERAPEUTIC COMPOSITIONS AND METHODS PFIZER (US) 1997-02-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050131040-A1 Process for the preparation of crystalline losartan potassium REN, AGT, ACE AGTR1 4/4885AGTR2 5/4885GP6 3713/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.