SCHEMBL4678735

SCHEMBL4678735

Nc1ccc(CN(C(=O)O)C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.38
MAPT P10636 1/20 0.37
ALDH1A1 P00352 3/20 0.37
GFER P55789 1/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MAOB P27338 4/20 0.36
MAOA P21397 2/20 0.36
CES1 P23141 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.35
TAS2R14 Q9NYV8 1/20 0.35
ITGB1 P05556 2/20 0.35
ITGA5 P08648 2/20 0.35
LMNA P02545 1/20 0.35
ITGB3 P05106 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250885 0.82 CES1 (0.53) ALDH1A1TDP1CES1MEN1KMT2A
SCHEMBL335254 0.81 MEN1 (0.50) FDPSMAPTALDH1A1GFERCYP3A4
SCHEMBL28614083 0.79 HDAC3 (0.37) MAPTALDH1A1MEN1KMT2AHTT
SCHEMBL10338250 0.74 MEN1 (0.46) ALDH1A1TDP1CES1MEN1KMT2A
SCHEMBL7306368 0.74 GFER (0.44) FDPSMAPTALDH1A1GFERCYP3A4
SCHEMBL6968790 0.73 KDM4E (0.47) MAPTALDH1A1TSHRTDP1MAOB
SCHEMBL24193442 0.72 MEN1 (0.47) ALDH1A1TDP1CES1MEN1KMT2A
SCHEMBL14269830 0.71 RIPK1 (0.50) MAPTALDH1A1TDP1MEN1KMT2A
SCHEMBL5007989 0.71 MEN1 (0.44) ALDH1A1TDP1CES1MEN1KMT2A
SCHEMBL4806015 0.71 RAB9A (0.50) MAPTALDH1A1MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957460-A1 BICYCLIC COMPOUNDS WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-08-20 EP disclosed
WO-2007067444-A1 BICYCLIC COMPOUNDS WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-06-14 WO disclosed