SCHEMBL4684089

SCHEMBL4684089

CCOC(=O)c1cc(F)cc(CC(C)(F)CC2CN(C(c3ccc(Cl)cc3)c3cccc(C#N)c3)C2)c1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.36
ELANE P08246 10/20 0.34
CNR1 P21554 7/20 0.34
CNR2 P34972 6/20 0.34
CYP2C9 P11712 2/20 0.34
KLKB1 P03952 1/20 0.34
CYP2D6 P10635 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4681581 0.95 ELANE (0.38) MGLLELANECYP2C9KLKB1
SCHEMBL4796795 0.91 ELANE (0.34) MGLLELANECYP2C9
SCHEMBL4683968 0.90 CNR1 (0.37) MGLLCNR1CNR2CYP2C9KLKB1
SCHEMBL4968374 0.88 CNR1 (0.39) MGLLCNR1CNR2CYP2C9KLKB1
SCHEMBL4080122 0.88 CNR1 (0.40) MGLLCNR1CNR2
SCHEMBL5727699 0.86 CNR1 (0.38) MGLLCNR1CNR2
SCHEMBL4684135 0.85 OPRD1 (0.41)
SCHEMBL4966303 0.84 MGLL (0.40) MGLLKLKB1
SCHEMBL4787427 0.84 CNR1 (0.36) MGLLCNR1CNR2KLKB1
SCHEMBL1500546 0.83 MGLL (0.37) MGLLELANECNR1CNR2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960392-A2 HETEROCYCLE-SUBSTITUTED 3-ALKYL AZETIDINE DERIVATIVES Merck & Co., Inc. (US) 2008-08-27 EP disclosed
WO-2007064566-A2 HETEROCYCLE-SUBSTITUTED 3-ALKYL AZETIDINE DERIVATIVES MERCK & CO., INC. (US) 2007-06-07 WO disclosed