SCHEMBL4684285

SCHEMBL4684285

OCCCCSc1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.44
CA2 P00918 2/20 0.42
ALDH1A1 P00352 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
TBXAS1 P24557 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
PLA2G7 Q13093 5/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 1/20 0.38
CLK1 P49759 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682354 0.98 CA2 (0.44) GRM2CA2ALDH1A1SMN1; SMN2NPC1
SCHEMBL4684945 0.98 CA2 (0.44) GRM2CA2ALDH1A1SMN1; SMN2NPC1
SCHEMBL4687467 0.95 ALDH1A1 (0.43) GRM2CA2ALDH1A1SMN1; SMN2NPC1
SCHEMBL4684826 0.87 MAPK1 (0.47) GRM2CA2ALDH1A1SMN1; SMN2NPC1
SCHEMBL4684282 0.82 GRM2 (0.44) GRM2ALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8429843 0.82 GRM2 (0.41) GRM2ALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8616038 0.82 GRM2 (0.44) GRM2ALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8427404 0.81 GRM2 (0.40) GRM2ALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL4682349 0.81 GRM2 (0.43) GRM2ALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL4684941 0.81 GRM2 (0.43) GRM2ALDH1A1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed