SCHEMBL4684945

SCHEMBL4684945

OCCCCCSc1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.44
TBXAS1 P24557 1/20 0.43
GRM2 Q14416 1/20 0.43
PLA2G7 Q13093 6/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682354 1.00 CA2 (0.44) CA2TBXAS1GRM2PLA2G7SMN1; SMN2
SCHEMBL4684285 0.98 GRM2 (0.44) CA2TBXAS1GRM2PLA2G7SMN1; SMN2
SCHEMBL4687467 0.93 ALDH1A1 (0.43) CA2TBXAS1GRM2SMN1; SMN2NPC1
SCHEMBL4684826 0.85 MAPK1 (0.47) CA2GRM2SMN1; SMN2NPC1RAB9A
SCHEMBL8427404 0.83 GRM2 (0.40) GRM2PLA2G7SMN1; SMN2NPC1RAB9A
SCHEMBL4682349 0.83 GRM2 (0.43) GRM2PLA2G7SMN1; SMN2NPC1RAB9A
SCHEMBL4684941 0.83 GRM2 (0.43) GRM2PLA2G7SMN1; SMN2NPC1RAB9A
SCHEMBL28082118 0.82 PLA2G7 (0.43) GRM2PLA2G7SMN1; SMN2NPC1RAB9A
SCHEMBL8616038 0.81 GRM2 (0.44) GRM2PLA2G7SMN1; SMN2NPC1RAB9A
SCHEMBL4684282 0.81 GRM2 (0.44) GRM2PLA2G7SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed
EP-0232623-B1 1-CARBACEPHALOSPORIN ANTIBIOTICS ELI LILLY AND COMPANY (US) 1993-03-17 EP disclosed
US-4892942-A 1-CARBA (DETHIA)CEPHALOSPORINS ELI LILLY AND COMPANY (US) 1990-01-09 US disclosed
US-4791106-A 1-Carbacephalosporin antibiotics ELI LILLY AND COMPANY (US) 1988-12-13 US disclosed
EP-0232623-A1 1-Carbacephalosporin antibiotics ELI LILLY AND COMPANY (US) 1987-08-19 EP disclosed