SCHEMBL4684596

SCHEMBL4684596

COc1c(COC(C)=O)ncc(Br)c1OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
THRB P10828 2/20 0.42
THRA P10827 1/20 0.42
KCNA3 P22001 1/20 0.41
PTPN1 P18031 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
PDE4D Q08499 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
MAOB P27338 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
BLM P54132 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4685977 0.80 THRA (0.46) THRBTHRAKCNA3MEN1KMT2A
SCHEMBL30468864 0.80 THRA (0.46) THRBTHRAKCNA3MEN1KMT2A
SCHEMBL6876891 0.79 ALDH1A1 (0.51) ALDH1A1KCNA3PTPN1HPGDPDE4D
SCHEMBL10247054 0.79 PTPN1 (0.55) ALDH1A1PTPN1LMNAHPGDSMN1; SMN2
SCHEMBL3799664 0.78 AGXT (0.44) ALDH1A1MEN1KMT2AMAPT
SCHEMBL4687273 0.78 ALDH1A1 (0.53) ALDH1A1KCNA3PTPN1HPGDSMN1; SMN2
SCHEMBL19755566 0.76 ALDH1A1 (0.48) ALDH1A1PTPN1MEN1KMT2ALMNA
SCHEMBL4681950 0.76 L3MBTL1 (0.42) ALDH1A1THRBTHRAMEN1KMT2A
SCHEMBL19625790 0.76 ALDH1A1 (0.50) ALDH1A1KCNA3PTPN1LMNAHPGD
SCHEMBL83012 0.75 ALDH1A1 (0.47) ALDH1A1PTPN1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973906-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE Virochem Pharma Inc. (CA) 2008-10-01 EP disclosed
WO-2006066414-A1 HYDROXYDIHYDROPYRIDOPY RAZINE-1,8-DIONES AND METHODS FOR INHIBITING HIV INTEGRASE VIROCHEM PHARMA INC. (CA) 2006-06-29 WO disclosed