SCHEMBL4685250

SCHEMBL4685250

CC(C[O])CSc1cnc[nH]1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 10/20 0.36
HRH4 Q9H3N8 9/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.36
GLA P06280 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1A2 P05177 1/20 0.36
NFKB1 P19838 1/20 0.36
THPO P40225 1/20 0.36
LMNA P02545 1/20 0.35
APEX1 P27695 1/20 0.35
BLM P54132 1/20 0.35
CPB1 P15086 1/20 0.33
CPB2 Q96IY4 1/20 0.33
FKBP5 Q13451 1/20 0.32
QPCT Q16769 1/20 0.32
QPCTL Q9NXS2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633118 0.83 PKM (0.37) HRH3HRH4ALDH1A1MEN1GLA
SCHEMBL8429888 0.79 HRH3 (0.38) HRH3HRH4ALDH1A1MEN1GLA
SCHEMBL7285552 0.68
SCHEMBL4683083 0.68 HRH3 (0.35) HRH3HRH4ALDH1A1MEN1KMT2A
SCHEMBL17368394 0.67
SCHEMBL7296375 0.67 HRH3 (0.35) HRH3HRH4ALDH1A1MEN1KMT2A
SCHEMBL4680899 0.66 MEN1 (0.38) HRH3ALDH1A1MEN1KMT2ACYP1A2
SCHEMBL4684977 0.64 ALDH1A1 (0.38) HRH3HRH4ALDH1A1MEN1GLA
SCHEMBL6169087 0.64 HRH3 (0.47) HRH3HRH4ALDH1A1CYP1A2LMNA
SCHEMBL10934277 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed