SCHEMBL4685646

SCHEMBL4685646

CCC1CCCCC1(O)c1ccccc1OC(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.46
TRPA1 O75762 4/20 0.37
SLC6A4 P31645 7/20 0.35
SLC6A2 P23975 5/20 0.35
SLC22A1 O15245 3/20 0.35
OPRM1 P35372 3/20 0.35
OPRD1 P41143 3/20 0.35
SLC6A3 Q01959 2/20 0.35
CHRM2 P08172 2/20 0.35
CHRM1 P11229 2/20 0.35
OPRK1 P41145 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM3 P20309 1/20 0.34
PDK2 Q15119 1/20 0.34
BACE1 P56817 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4984839 0.84 CHRM2 (0.49) SLC6A4SLC6A2SLC22A1OPRM1OPRD1
SCHEMBL4991842 0.81 HDAC4 (0.44) TRPA1SLC6A4SLC6A2SLC22A1OPRM1
SCHEMBL6470509 0.80 SLC6A9 (0.37) SLC6A9BACE1CYP3A4CYP2C19
SCHEMBL4540371 0.79 MEN1 (0.42) SLC6A4SLC6A2OPRM1OPRD1SLC6A3
SCHEMBL4989694 0.72 SLC6A2 (0.51) SLC6A9SLC6A4SLC6A2SLC22A1OPRM1
SCHEMBL6865381 0.71 SLC6A2 (0.60) SLC6A4SLC6A2SLC22A1OPRM1OPRD1
SCHEMBL5695493 0.70 HDAC4 (0.40) SLC6A4SLC6A2PDK2
SCHEMBL4685654 0.70 HCRTR2 (0.36) SLC6A9TRPA1SLC6A4SLC6A3CYP3A4
Hydrochloric Acid SCHEMBL8686122 0.70 SLC6A2 (0.59) SLC6A4SLC6A2SLC22A1OPRM1OPRD1
SCHEMBL5718315 0.68 SLC6A2 (0.44) SLC6A4SLC6A2SLC22A1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957470-A1 PROCESS FOR SELECTIVE SYNTHESIS OF ENANTIOMERS OF SUBSTITUTED 1-(2-AMINO-1-PHENYL-ETHYL)-CYCLOHEXANOLS Wyeth (US) 2008-08-20 EP disclosed
WO-2007067501-A1 PROCESS FOR SELECTIVE SYNTHESIS OF ENANTIOMERS OF SUBSTITUTED 1-(2-AMINO-1-PHENYL-ETHYL)-CYCLOHEXANOLS WYETH (US) 2007-06-14 WO disclosed
EP-1673059-A2 ALKANOL AND CYCLOALKANOL-AMINE DERIVATIVES AND METHODS OF THEIR USE Wyeth (US) 2006-06-28 EP disclosed
EP-1673090-A1 FUSED-ARYL AND HETEROARYL DERIVATIVES AND METHODS OF THEIR USE Wyeth (US) 2006-06-28 EP disclosed
WO-2005037207-A2 ARYLALKYL-PIPERAZINE DERIVATIVES FOR THE TREATMENT OF CONDITIONS AMELIORATED BY MONOAMINE REUPTAKE INCLUDING VASOMOTOR SYMPTOMS (VMS) WYETH (US) 2005-04-28 WO disclosed
WO-2005037283-A1 FUSED-ARYL AND HETEROARYL DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2005-04-28 WO disclosed