SCHEMBL4686158

SCHEMBL4686158

OCc1ccn(-c2ccc(-c3cc(CNc4ccon4)on3)cc2F)c1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.33
NOTUM Q6P988 2/20 0.32
POLB P06746 1/20 0.30
JAK2 O60674 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4679245 0.85 IGF1R (0.34) IGF1R
SCHEMBL4686151 0.84 IGF1R (0.33) IGF1RPOLBALDH1A1
SCHEMBL4683030 0.84 IGF1R (0.33) IGF1RPOLB
SCHEMBL4679791 0.82 BLM (0.37) IGF1R
SCHEMBL14066488 0.80 PSEN1 (0.43) IGF1R
SCHEMBL3582885 0.78 IGF1R (0.46) IGF1RNOTUMPOLBJAK2ALDH1A1
SCHEMBL4680635 0.78 IGF1R (0.32) IGF1R
SCHEMBL3591482 0.76 IGF1R (0.40) IGF1R
SCHEMBL4679278 0.75 IGF1R (0.37) IGF1RNOTUMPOLBJAK2ALDH1A1
SCHEMBL4682699 0.73 GAA (0.38) POLBJAK2ALDH1A1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1437349-B9 SUBSTITUTED ISOXAZOLES AND THE USE THEREOF AS ANTIBIOTICS S A L V A T LAB SA (ES) 2008-09-10 EP disclosed
EP-1437349-B1 SUBSTITUTED ISOXAZOLES AND THE USE THEREOF AS ANTIBIOTICS S A L V A T LAB SA (ES) 2007-08-15 EP disclosed
US-20050014806-A1 Substituted isoxazoles and their use as antibiotics LABORATORIOS S.A.L.V.A.T., S.A. (ES) 2005-01-20 US disclosed
EP-1437349-A1 SUBSTITUTED ISOXAZOLES AND THE USE THEREOF AS ANTIBIOTICS LABORATORIOS S.A.L.V.A.T., S.A. (ES) 2004-07-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014806-A1 Substituted isoxazoles and their use as antibiotics XDH, SCO2, HAX1 IGF1R 798/4885NOTUM 3353/4885POLB 1162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.