SCHEMBL4687638

SCHEMBL4687638

CN1CCOc2cc([S+]([O-])n3nc(N4CCNCC4)c4ccccc43)ccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.36
NOTUM Q6P988 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
ALOX15 P16050 1/20 0.34
LCK P06239 1/20 0.34
TNK2 Q07912 1/20 0.34
PTGES2 Q9H7Z7 1/20 0.33
TRPM5 Q9NZQ8 1/20 0.33
PDE10A Q9Y233 1/20 0.33
KDM1A O60341 2/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
METAP2 P50579 1/20 0.32
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4744859 0.81 KDR (0.35) GBA1NOTUMCYP11B1CYP11B2ALDH1A1
SCHEMBL3339496 0.78 GBA1 (0.49) GBA1NOTUMALDH1A1PTGES2SCN5A
SCHEMBL4741748 0.76 CYP11B1 (0.34) CYP11B1CYP11B2ALOX15PTGES2TRPM5
SCHEMBL3337670 0.68 GBA1 (0.54) GBA1ALDH1A1CYP3A4CYP2D6PTGES2
SCHEMBL3339265 0.68 HTR6 (0.51) GBA1CYP3A4CYP2D6PTGES2
SCHEMBL30643702 0.66 DDB1 (0.52) CYP1A2CYP3A4CYP2D6ADRB2ADRB1
SCHEMBL2710143 0.66 DDB1 (0.52) CYP1A2CYP3A4CYP2D6ADRB2ADRB1
SCHEMBL3644217 0.64 HTR6 (0.62)
SCHEMBL5095027 0.62 KHK (0.45) GBA1NOTUMALDH1A1PTGES2HTT
SCHEMBL18903778 0.61 CYP11B1 (0.39) NOTUMCYP11B1CYP11B2ALDH1A1PTGES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984351-A1 COMPOUNDS HAVING 5-HT6 RECEPTOR AFFINITY Memory Pharmaceuticals Corporation (US) 2008-10-29 EP disclosed
WO-2007098418-A1 COMPOUNDS HAVING 5-HT6 RECEPTOR AFFINITY MEMORY PHARMACEUTICALS CORPORATION (US) 2007-08-30 WO disclosed