SCHEMBL4688433

SCHEMBL4688433

Cc1cc(Cl)ccc1-c1cc(F)cc2c1O[C]C2

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.43
NOTUM Q6P988 2/20 0.35
MAPK14 Q16539 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047914 0.82 S1PR1 (0.34) AQP1
SCHEMBL4596881 0.81 NOTUM (0.36) NOTUMMAPK14
SCHEMBL4764345 0.75 AQP1 (0.56) AQP1NOTUMMAPK14
SCHEMBL4764341 0.74 AQP1 (0.55) AQP1NOTUMMAPK14
SCHEMBL4226033 0.72 AQP1 (0.80) AQP1NOTUMMAPK14
SCHEMBL4229976 0.72 AQP1 (0.62) AQP1NOTUM
SCHEMBL5605280 0.72 AQP1 (0.58) AQP1NOTUM
SCHEMBL4229969 0.72 AQP1 (0.62) AQP1NOTUM
SCHEMBL14113467 0.72 AQP1 (0.80) AQP1NOTUMMAPK14
SCHEMBL28760844 0.70 AQP1 (0.60) AQP1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
WO-2007030150-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH (US) 2007-03-15 WO disclosed