SCHEMBL4690403

SCHEMBL4690403

Cc1cc(Cl)c(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.39
HCRTR2 O43614 8/20 0.39
TNF P01375 1/20 0.38
CCR5 P51681 5/20 0.36
TACR1 P25103 1/20 0.35
S1PR1 P21453 1/20 0.34
HPGD P15428 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694334 0.94 HCRTR1 (0.43) HCRTR1HCRTR2TNFCCR5TACR1
SCHEMBL4693010 0.91 HCRTR1 (0.36) HCRTR1HCRTR2TNFCCR5TACR1
SCHEMBL3281863 0.90 HCRTR1 (0.48) HCRTR1HCRTR2TNFCCR5
SCHEMBL4695961 0.90 HCRTR1 (0.36) HCRTR1HCRTR2TNFCCR5
SCHEMBL3283594 0.87 CCL5 (0.43) CCR5
SCHEMBL4694815 0.87 HCRTR1 (0.37) HCRTR1HCRTR2TNFCCR5PDE4B
SCHEMBL4694788 0.87 HCRTR1 (0.45) HCRTR1HCRTR2TNFCCR5
SCHEMBL4695935 0.87 HCRTR2 (0.47) HCRTR1HCRTR2TNFHPGDALDH1A1
SCHEMBL4694763 0.87 HCRTR1 (0.37) HCRTR1HCRTR2TNFCCR5PDE4B
SCHEMBL4695956 0.87 HCRTR1 (0.37) HCRTR1HCRTR2TNFCCR5S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed