SCHEMBL4690501

SCHEMBL4690501

COc1ccc(-n2nc(C)cc2C(=O)N2CC3CN(CC[C@H](N)c4ccccc4)CC3C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
CCR5 P51681 5/20 0.45
F10 P00742 3/20 0.41
ADRB1 P08588 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2B P41595 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
DHODH Q02127 1/20 0.41
CCL5 P13501 2/20 0.40
LMNA P02545 2/20 0.40
GFER P55789 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 2/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690543 0.83 CCR5 (0.46) TSHRCCR5CCL5ALDH1A1
SCHEMBL4690555 0.81 MAPK14 (0.52) CCR5ADRB1HTR2AHTR2BSIGMAR1
SCHEMBL4692822 0.81 SMYD3 (0.46) CCR5CCL5ALDH1A1HTT
SCHEMBL4691481 0.79 CCR5 (0.49) TSHRCCR5
SCHEMBL4690568 0.79 CCR5 (0.67) CCR5CCL5
SCHEMBL4691935 0.78 KDM4E (0.42) CCR5ADRB1HTR2AHTR2BSIGMAR1
SCHEMBL4694118 0.77 KCNK3 (0.51) CCR5MEN1KMT2AALDH1A1
SCHEMBL4690598 0.77 CCR5 (0.55) CCR5CCL5
SCHEMBL4690500 0.76 F10 (0.43) TSHRF10ADRB1HTR2AHTR2B
SCHEMBL4695964 0.76 CCR5 (0.54) CCR5CCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed