SCHEMBL4690543

SCHEMBL4690543

Cc1cc(C(=O)N2CC3CN(CC[C@H](N)c4ccccc4)CC3C2)n(C)n1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 11/20 0.46
CCL5 P13501 10/20 0.45
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692822 0.89 SMYD3 (0.46) CCR5CCL5ALDH1A1
SCHEMBL4690462 0.88 MEN1 (0.46) CCR5CCL5ALDH1A1
Cyclopentane SCHEMBL4694432 0.85 CCR5 (0.58) CCR5
SCHEMBL4690501 0.83 TSHR (0.49) CCR5CCL5ALDH1A1TSHR
SCHEMBL4693123 0.81 CCR5 (0.50) CCR5CCL5ALDH1A1
SCHEMBL4696493 0.80 CCR5 (0.59) CCR5CCL5
SCHEMBL4694458 0.80 CCR5 (0.53) CCR5CCL5
SCHEMBL4694095 0.79 CCR5 (0.51) CCR5CCL5
SCHEMBL3290682 0.79 CCR5 (0.70) CCR5CCL5
SCHEMBL3285413 0.79 CCR5 (0.70) CCR5CCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed