SCHEMBL4690500

SCHEMBL4690500

COc1ccc(-n2nc(C(N)=O)cc2C(=O)N2CC3CN(CC[CH]c4ccccc4)C[C@H]3C2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
F10 P00742 6/20 0.43
KLKB1 P03952 1/20 0.43
DHODH Q02127 5/20 0.41
F5 P12259 1/20 0.39
BRSK2 Q8IWQ3 1/20 0.39
RPA1 P27694 1/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
FAAH O00519 1/20 0.38
MGLL Q99685 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 1/20 0.38
ADRB1 P08588 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2B P41595 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690538 0.84 CCL5 (0.36)
SCHEMBL4692820 0.82 CCL5 (0.35) ALDH1A1HTT
SCHEMBL4690567 0.77 CCR5 (0.51)
SCHEMBL4690501 0.76 TSHR (0.49) F10DHODHALDH1A1LMNAHTT
SCHEMBL4690594 0.74 CCR5 (0.44)
SCHEMBL4692504 0.74 HCRTR1 (0.44) ALDH1A1LMNA
SCHEMBL4690551 0.73 MAPK14 (0.41) ALDH1A1LMNA
SCHEMBL4690459 0.73 MEN1 (0.37) ALDH1A1
SCHEMBL4694094 0.73 CHRNB2 (0.44) ALDH1A1L3MBTL1
SCHEMBL4690761 0.72 KDM4E (0.43) ALDH1A1LMNAHTTL3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed