SCHEMBL4690504

SCHEMBL4690504

COc1cc(Cl)ccc1C(=O)N1CC2CN(CCCNC(=O)c3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.50
HCRTR2 O43614 1/20 0.50
F10 P00742 2/20 0.48
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
DRD2 P14416 6/20 0.45
DRD4 P21917 5/20 0.45
DRD3 P35462 4/20 0.45
HTR4 Q13639 1/20 0.44
DRD1 P21728 1/20 0.44
KMT2A Q03164 1/20 0.42
CCR3 P51677 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
SLC29A1 Q99808 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691870 0.93 F10 (0.50) F10CYP2D6CYP2C9DRD2DRD4
SCHEMBL4690666 0.91 NTRK1 (0.44) HCRTR1HCRTR2F10DRD2DRD4
SCHEMBL4694269 0.89 HCRTR1 (0.48) HCRTR1HCRTR2F10DRD2DRD4
SCHEMBL4690744 0.88 NTRK1 (0.42) HCRTR1HCRTR2F10DRD2DRD4
SCHEMBL4690506 0.86 HCRTR1 (0.52) HCRTR1HCRTR2
SCHEMBL4696371 0.84 TSHR (0.44) CYP2C9
SCHEMBL4693332 0.84 SLC6A4 (0.45) DRD2DRD4DRD3
SCHEMBL4691666 0.84 CCR3 (0.47) F10CYP2D6CYP2C9DRD2DRD4
SCHEMBL4695945 0.84 NTRK1 (0.44) HCRTR1HCRTR2F10CYP2C9DRD2
SCHEMBL4692993 0.83 TSHR (0.43) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed