SCHEMBL4690744

SCHEMBL4690744

Cc1ccc(C(=O)NCCCN2CC3CN(C(=O)c4ccc(Cl)cc4F)CC3C2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.42
MAPT P10636 1/20 0.41
KMT2A Q03164 2/20 0.41
SLC6A4 P31645 1/20 0.41
LMNA P02545 2/20 0.40
TMEM97 Q5BJF2 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
F10 P00742 1/20 0.40
MAPK14 Q16539 1/20 0.40
GAA P10253 1/20 0.40
MEN1 O00255 1/20 0.40
CACNA1G O43497 1/20 0.40
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CCR1 P32246 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690666 0.93 NTRK1 (0.44) NTRK1MAPTKMT2ASLC6A4LMNA
SCHEMBL4694269 0.91 HCRTR1 (0.48) NTRK1MAPTKMT2ASLC6A4LMNA
SCHEMBL4695321 0.89 TSHR (0.43) MAPTLMNASMN1; SMN2MAPK14
SCHEMBL4694433 0.89 P2RX7 (0.45) MAPTKMT2ALMNASMN1; SMN2MAPK14
SCHEMBL4690504 0.88 HCRTR1 (0.50) KMT2AF10HCRTR1HCRTR2DRD2
SCHEMBL4694384 0.87 SLC6A4 (0.42) KMT2ASLC6A4LMNASMN1; SMN2MEN1
SCHEMBL4692216 0.87 SLC6A2 (0.43) SLC6A4LMNASMN1; SMN2MAPK14GAA
SCHEMBL4695512 0.87 LMNA (0.41) NTRK1KMT2ASLC6A4LMNATMEM97
SCHEMBL4690747 0.86 HCRTR1 (0.41) MAPTLMNASMN1; SMN2GAAHCRTR1
SCHEMBL4691870 0.86 F10 (0.50) KMT2ASMN1; SMN2F10MEN1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed