SCHEMBL4695945

SCHEMBL4695945

Cc1ccc(C(=O)NCCCN2CC3CN(C(=O)c4cc(Cl)ccc4-n4c(C)ccc4C)CC3C2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.44
HCRTR1 O43613 3/20 0.42
HCRTR2 O43614 3/20 0.42
MAPT P10636 1/20 0.41
F10 P00742 1/20 0.41
SLC6A4 P31645 2/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
MAPK14 Q16539 1/20 0.40
CACNA1G O43497 2/20 0.40
DRD2 P14416 3/20 0.39
DRD3 P35462 3/20 0.39
DRD4 P21917 2/20 0.39
GSK3B P49841 1/20 0.39
MYC P01106 1/20 0.39
NR4A1 P22736 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694269 0.90 HCRTR1 (0.48) NTRK1HCRTR1HCRTR2MAPTF10
SCHEMBL4690666 0.89 NTRK1 (0.44) NTRK1HCRTR1HCRTR2MAPTF10
SCHEMBL4691870 0.87 F10 (0.50) F10DRD2DRD3DRD4CYP2C9
SCHEMBL4695946 0.86 HCRTR1 (0.43) HCRTR1HCRTR2MAPTMYCNR4A1
SCHEMBL4690744 0.85 NTRK1 (0.42) NTRK1HCRTR1HCRTR2MAPTF10
SCHEMBL4690504 0.84 HCRTR1 (0.50) HCRTR1HCRTR2F10DRD2DRD3
SCHEMBL4693332 0.83 SLC6A4 (0.45) SLC6A4DRD2DRD3DRD4
SCHEMBL4691761 0.83 SLC6A2 (0.44) SLC6A4MAPK14DRD2DRD3DRD4
SCHEMBL3284096 0.82 SMYD2 (0.44) SLC6A4MAPK14DRD2DRD3DRD4
SCHEMBL4690664 0.82 SMYD2 (0.43) MAPTSLC6A4MAPK14DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed