SCHEMBL4690649

SCHEMBL4690649

Cc1ccc(NCC(O)CN2CC3CN(C(=O)c4c(C)ccnc4C)CC3C2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 13/20 0.47
CCL5 P13501 11/20 0.39
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3283296 0.88 CCR5 (0.48) CCR5MAPTHTT
SCHEMBL4693868 0.87 CCR5 (0.48) CCR5CCL5HTT
SCHEMBL4694037 0.84 MALT1 (0.42) CCR5MAPTHTT
SCHEMBL3282227 0.84 CCR5 (0.51) CCR5CCL5KCNH2
SCHEMBL3283576 0.81 CCR5 (0.44) CCR5CCL5MAPTKCNH2
SCHEMBL3282221 0.80 CCR5 (0.51) CCR5CCL5MAPTHTT
SCHEMBL4692314 0.80 LMNA (0.45) MAPTHTT
SCHEMBL13359815 0.80 CCR5 (0.50) CCR5KCNH2
SCHEMBL3283988 0.79 CCR5 (0.48) CCR5MAPTHTT
SCHEMBL4693629 0.79 CCR5 (0.51) CCR5CCL5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed