SCHEMBL4690883

SCHEMBL4690883

Cc1ccc(NCCCN2CC3CN(S(=O)(=O)c4cnn(-c5ccccc5)c4C)CC3C2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.41
ALDH1A1 P00352 5/20 0.39
MAPT P10636 4/20 0.39
TP53 P04637 4/20 0.39
SMN1; SMN2 Q16637 5/20 0.38
POLB P06746 1/20 0.38
GAA P10253 3/20 0.38
AGTR1 P30556 1/20 0.38
KDM4E B2RXH2 2/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691686 0.85 MAPT (0.48) NR1H4ALDH1A1MAPTTP53SMN1; SMN2
SCHEMBL4690880 0.84 TP53 (0.50) NR1H4ALDH1A1MAPTTP53SMN1; SMN2
SCHEMBL3283683 0.81 MAPT (0.47) ALDH1A1MAPTTP53SMN1; SMN2GAA
SCHEMBL4691706 0.80 MAPT (0.47) NR1H4ALDH1A1MAPTTP53SMN1; SMN2
SCHEMBL4691506 0.79 NR1H4 (0.49) NR1H4ALDH1A1MAPTTP53SMN1; SMN2
SCHEMBL3283552 0.79 CCR1 (0.42) ALDH1A1MAPTTP53SMN1; SMN2GAA
SCHEMBL4695133 0.79 NR1H4 (0.46) NR1H4ALDH1A1MAPTTP53SMN1; SMN2
SCHEMBL4691665 0.78 TP53 (0.41) ALDH1A1MAPTTP53SMN1; SMN2POLB
SCHEMBL4694266 0.78 MAPT (0.46) ALDH1A1MAPTTP53SMN1; SMN2GAA
SCHEMBL4692449 0.77 ALDH1A1 (0.46) ALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed