SCHEMBL4691722

SCHEMBL4691722

Cc1ccc(N(CCCN2CC3=CN(C(=O)c4c(C)ccnc4C)CC3C2)C(=O)Nc2cccc(Cl)c2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 5/20 0.39
UBE2M P61081 2/20 0.35
DCUN1D1 Q96GG9 2/20 0.35
MAPT P10636 3/20 0.34
HSD17B10 Q99714 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
TSHR P16473 2/20 0.34
KDM4E B2RXH2 2/20 0.34
USP2 O75604 2/20 0.34
TP53 P04637 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
PKM P14618 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MCHR1 Q99705 4/20 0.34
KCNH2 Q12809 3/20 0.33
USP30 Q70CQ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694952 0.94 CCR5 (0.37) CCR5UBE2MDCUN1D1LMNAKCNH2
SCHEMBL4690445 0.92 EPHX2 (0.38) CCR5KCNH2
SCHEMBL4691638 0.92 CCR5 (0.37) CCR5MCHR1KCNH2
SCHEMBL4690611 0.91 CCR5 (0.37) CCR5UBE2MDCUN1D1MAPTKCNH2
SCHEMBL4694148 0.90 MAPT (0.36) CCR5UBE2MDCUN1D1MAPTTP53
SCHEMBL4691621 0.90 CCR5 (0.35) CCR5KCNH2
SCHEMBL4690740 0.90 CCR5 (0.42) CCR5KCNH2
SCHEMBL4694359 0.90 CCR5 (0.34) CCR5UBE2MDCUN1D1KCNH2USP30
SCHEMBL4695361 0.89 CCR5 (0.37) CCR5KCNH2
SCHEMBL4694995 0.89 CCR5 (0.34) CCR5MCHR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed