SCHEMBL4691744

SCHEMBL4691744

Cc1ccc(C(=O)NCCCN2CC3CN(C(=O)c4cc5ccccc5s4)CC3C2)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.51
SLC6A2 P23975 4/20 0.51
DRD2 P14416 11/20 0.50
DRD3 P35462 9/20 0.50
DRD4 P21917 3/20 0.50
HTR1A P08908 2/20 0.48
DRD1 P21728 2/20 0.48
ADRA1D P25100 2/20 0.48
HTR2A P28223 2/20 0.48
HTR2C P28335 2/20 0.48
ADRA1A P35348 2/20 0.48
ADRA1B P35368 2/20 0.48
HTR2B P41595 2/20 0.48
HRH4 Q9H3N8 1/20 0.45
RAB9A P51151 1/20 0.44
CCR1 P32246 1/20 0.43
ACKR3 P25106 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691748 0.86 HRH4 (0.46) SLC6A4SLC6A2DRD2DRD3DRD4
SCHEMBL4691639 0.85 SMYD2 (0.48) SLC6A4SLC6A2DRD2DRD3DRD4
SCHEMBL4693332 0.83 SLC6A4 (0.45) SLC6A4SLC6A2DRD2DRD3DRD4
SCHEMBL4690664 0.82 SMYD2 (0.43) SLC6A4SLC6A2DRD2DRD3DRD4
SCHEMBL4692849 0.82 DRD3 (0.49) SLC6A4SLC6A2DRD2DRD3DRD4
SCHEMBL4691221 0.81 L3MBTL3 (0.45)
SCHEMBL4693959 0.81 HCRTR1 (0.45) SLC6A4SLC6A2DRD2DRD3DRD4
SCHEMBL4691761 0.81 SLC6A2 (0.44) SLC6A4SLC6A2DRD2DRD3DRD4
SCHEMBL4691509 0.81 CCR5 (0.51) SLC6A4SLC6A2DRD2DRD3DRD4
SCHEMBL4692672 0.80 SMYD2 (0.45) SLC6A4SLC6A2DRD2DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed