SCHEMBL4691783

SCHEMBL4691783

NC(=O)c1c(F)cccc1C(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.41
HCRTR2 O43614 12/20 0.41
SLC6A1 P30531 3/20 0.37
CCR5 P51681 3/20 0.37
KCNK3 O14649 2/20 0.36
KCNK9 Q9NPC2 2/20 0.36
CYP1A2 P05177 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694116 0.86 HCRTR2 (0.38) HCRTR1HCRTR2CCR5
SCHEMBL4690347 0.83 HCRTR2 (0.42) HCRTR1HCRTR2CCR5
SCHEMBL4691301 0.82 HCRTR1 (0.44) HCRTR1HCRTR2CCR5CYP1A2
SCHEMBL4695880 0.82 CCR5 (0.40) HCRTR1HCRTR2SLC6A1CCR5
SCHEMBL4690783 0.82 CCR5 (0.47) HCRTR1HCRTR2SLC6A1CCR5
SCHEMBL3290678 0.82 CCR5 (0.50) HCRTR1HCRTR2CCR5
SCHEMBL3285409 0.82 CCR5 (0.50) HCRTR1HCRTR2CCR5
SCHEMBL4692504 0.82 HCRTR1 (0.44) HCRTR1HCRTR2CCR5
SCHEMBL4691191 0.82 HCRTR1 (0.40) HCRTR1HCRTR2KCNK3KCNK9
SCHEMBL4694094 0.80 CHRNB2 (0.44) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed