SCHEMBL4691301

SCHEMBL4691301

NC(=O)c1ccccc1[CH]CCN1CC2CN(C(=O)c3c(F)cccc3F)C[C@@H]2C1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 14/20 0.44
HCRTR2 O43614 14/20 0.44
HTT P42858 1/20 0.38
CCR5 P51681 3/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3284141 0.93 CCR5 (0.42) HCRTR1HCRTR2CCR5
SCHEMBL4691673 0.91 HCRTR1 (0.38) HCRTR1HCRTR2CCR5
SCHEMBL4691802 0.88 CCR5 (0.48) HCRTR1HCRTR2CCR5
SCHEMBL4691928 0.87 MAPK1 (0.41) HCRTR1HCRTR2
SCHEMBL4694455 0.85 CHRNB2 (0.44) CCR5
SCHEMBL4690210 0.84 RBP4 (0.35) HCRTR1HCRTR2CCR5CYP2C9CYP2C19
SCHEMBL4689903 0.83 P2RX7 (0.41) HTTCCR5LMNACYP2C9CYP2C19
SCHEMBL4694309 0.83 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL4691783 0.82 HCRTR1 (0.41) HCRTR1HCRTR2CCR5CYP1A2
SCHEMBL4693059 0.81 CCR5 (0.37) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed