SCHEMBL4694352

SCHEMBL4694352

Cc1ccc(NC(=O)CCN2CC3CN(C(=O)c4cccc(Cl)c4Cl)CC3C2)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.47
F2R P25116 1/20 0.47
TP53 P04637 1/20 0.45
LMNA P02545 4/20 0.44
ALDH1A1 P00352 3/20 0.44
HSD17B10 Q99714 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
USP2 O75604 1/20 0.44
GAA P10253 1/20 0.44
P2RX7 Q99572 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691866 0.91 KMT2A (0.47) KMT2ATP53LMNAALDH1A1HPGD
SCHEMBL4692884 0.90 LMNA (0.48) KMT2ATP53LMNAALDH1A1HSD17B10
SCHEMBL4694022 0.89 P2RX7 (0.47) KMT2AP2RX7
SCHEMBL4694161 0.88 KMT2A (0.48) KMT2ATP53LMNAALDH1A1HPGD
SCHEMBL4691299 0.88 MAPT (0.49) KMT2ATP53LMNAHSD17B10HPGD
SCHEMBL4695646 0.88 KMT2A (0.48) KMT2ATP53LMNAALDH1A1HPGD
SCHEMBL4693483 0.88 HCRTR1 (0.48) KMT2AF2RTP53LMNAALDH1A1
SCHEMBL4694219 0.88 LMNA (0.46) KMT2ATP53LMNAALDH1A1HPGD
SCHEMBL4691903 0.88 MEN1 (0.55) KMT2ATP53LMNAALDH1A1MAPK1
SCHEMBL3281859 0.87 CCR5 (0.52) KMT2ATP53LMNAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed