SCHEMBL4692848

SCHEMBL4692848

NC(=O)C(=O)N1CCC(C(=O)N2CC3CN(CC[CH]c4ccccc4)C[C@H]3C2)CC1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
HPGD P15428 2/20 0.39
KMT2A Q03164 6/20 0.38
MEN1 O00255 4/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 2/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
POLB P06746 1/20 0.38
CCL5 P13501 1/20 0.37
CCR5 P51681 1/20 0.37
USP2 O75604 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692781 0.88 PKM (0.36) ALDH1A1HPGDKMT2AMEN1TSHR
SCHEMBL4694943 0.78 NPC1 (0.34) ALDH1A1KMT2ACA12CA1CA2
SCHEMBL4695377 0.77 CCR5 (0.37) TSHRCCL5CCR5
SCHEMBL4694094 0.75 CHRNB2 (0.44) ALDH1A1HPGDCA12CA1CA2
SCHEMBL4694111 0.75 KMT2A (0.34) ALDH1A1KDM4EKMT2ACCR5
SCHEMBL4693059 0.75 CCR5 (0.37) ALDH1A1KDM4EKMT2AMEN1CCL5
SCHEMBL4694116 0.74 HCRTR2 (0.38) CCR5
SCHEMBL4694056 0.74 PREP (0.41) ALDH1A1KMT2AMEN1
SCHEMBL4692061 0.73 CCR5 (0.37) ALDH1A1SMN1; SMN2CCL5CCR5
SCHEMBL4694498 0.73 CCR5 (0.37) CCL5CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed