SCHEMBL4692944

SCHEMBL4692944

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4ccc(F)cc4F)CC3C2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.41
HCRTR2 O43614 4/20 0.41
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
DPP4 P27487 1/20 0.39
CPS1 P31327 2/20 0.39
ALDH1A1 P00352 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MAPK14 Q16539 1/20 0.38
P2RX7 Q99572 4/20 0.37
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KCNK3 O14649 1/20 0.36
KCNK9 Q9NPC2 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692712 0.93 HCRTR1 (0.43) HCRTR1HCRTR2ALDH1A1P2RX7KCNK3
SCHEMBL4692703 0.93 HCRTR1 (0.48) HCRTR1HCRTR2ALDH1A1P2RX7KCNK3
SCHEMBL4693718 0.91 TSHR (0.38) HCRTR1HCRTR2DPP4SMN1; SMN2
SCHEMBL4691904 0.90 HCRTR1 (0.46) HCRTR1HCRTR2ALDH1A1KCNK3KCNK9
SCHEMBL4692106 0.90 HCRTR1 (0.50) HCRTR1HCRTR2P2RX7KCNK3KCNK9
SCHEMBL4694969 0.89 HCRTR1 (0.38) HCRTR1HCRTR2DPP4P2RX7KCNK3
SCHEMBL4694815 0.89 HCRTR1 (0.37) HCRTR1HCRTR2DPP4
SCHEMBL4691612 0.89 KDM1A (0.38) ALDH1A1MAPK1SMN1; SMN2KMT2A
SCHEMBL4694083 0.88 TSHR (0.40) HCRTR1HCRTR2DPP4ALDH1A1SMN1; SMN2
SCHEMBL4693169 0.88 HCRTR1 (0.50) HCRTR1HCRTR2P2RX7KCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed