SCHEMBL4693718

SCHEMBL4693718

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4cc(F)c(F)cc4F)CC3C2)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
HPGD P15428 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MGLL Q99685 2/20 0.36
TNF P01375 1/20 0.36
HCRTR1 O43613 10/20 0.36
HCRTR2 O43614 10/20 0.36
MAPT P10636 1/20 0.34
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694083 0.92 TSHR (0.40) TSHRHPGDSMN1; SMN2TNFHCRTR1
SCHEMBL4692712 0.91 HCRTR1 (0.43) MGLLTNFHCRTR1HCRTR2MAPT
SCHEMBL4694375 0.91 HCRTR1 (0.40) TSHRHPGDMGLLTNFHCRTR1
SCHEMBL4692944 0.91 HCRTR1 (0.41) SMN1; SMN2HCRTR1HCRTR2DPP4
SCHEMBL4691904 0.90 HCRTR1 (0.46) TSHRTNFHCRTR1HCRTR2MAPT
SCHEMBL4694969 0.89 HCRTR1 (0.38) TSHRHPGDTNFHCRTR1HCRTR2
SCHEMBL4692703 0.89 HCRTR1 (0.48) MGLLTNFHCRTR1HCRTR2
SCHEMBL4695647 0.88 HCRTR1 (0.48) TNFHCRTR1HCRTR2
SCHEMBL4694165 0.88 HCRTR1 (0.48) HPGDTNFHCRTR1HCRTR2
SCHEMBL4691612 0.87 KDM1A (0.38) SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed