SCHEMBL4694083

SCHEMBL4694083

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4cc(F)c(Cl)cc4Cl)CC3C2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
HPGD P15428 5/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 1/20 0.35
TNF P01375 1/20 0.35
HCRTR1 O43613 8/20 0.35
HCRTR2 O43614 8/20 0.35
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693718 0.92 TSHR (0.38) TSHRHPGDSMN1; SMN2MAPTTNF
SCHEMBL4696912 0.89 TNF (0.34) TSHRHPGDSMN1; SMN2TNFHCRTR1
SCHEMBL4691904 0.89 HCRTR1 (0.46) TSHRMAPTTNFHCRTR1HCRTR2
SCHEMBL4692712 0.88 HCRTR1 (0.43) MAPTTNFHCRTR1HCRTR2ALDH1A1
SCHEMBL4694969 0.88 HCRTR1 (0.38) TSHRHPGDTNFHCRTR1HCRTR2
SCHEMBL4694375 0.88 HCRTR1 (0.40) TSHRHPGDMAPTTNFHCRTR1
SCHEMBL4692944 0.88 HCRTR1 (0.41) SMN1; SMN2HCRTR1HCRTR2DPP4ALDH1A1
SCHEMBL4692703 0.88 HCRTR1 (0.48) TNFHCRTR1HCRTR2ALDH1A1
SCHEMBL4695647 0.87 HCRTR1 (0.48) TNFHCRTR1HCRTR2
SCHEMBL4694165 0.87 HCRTR1 (0.48) HPGDTNFHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed