SCHEMBL4693014

SCHEMBL4693014

Cc1cc(Cl)c(C(=O)N2CC3CN(CCCNc4ccc(C)c(Cl)c4)CC3C2)c(N2CCCC2)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
POLB P06746 2/20 0.41
TP53 P04637 1/20 0.41
CCR5 P51681 6/20 0.39
HTT P42858 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 3/20 0.37
USP2 O75604 1/20 0.37
MCL1 Q07820 1/20 0.37
AVPR2 P30518 2/20 0.36
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36
FKBP1A P62942 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690404 0.91 CCR5 (0.41) MAPTSMN1; SMN2POLBTP53CCR5
SCHEMBL4694337 0.87 CCR5 (0.43) MAPTSMN1; SMN2CCR5HTTL3MBTL1
SCHEMBL4693007 0.86 HTT (0.43) MAPTSMN1; SMN2TP53HTTL3MBTL1
SCHEMBL3281865 0.84 CCR5 (0.52) MAPTSMN1; SMN2CCR5HTTLMNA
SCHEMBL4695962 0.82 MEN1 (0.41) MAPTSMN1; SMN2CCR5HTTL3MBTL1
SCHEMBL4691511 0.82 CCR5 (0.54) MAPTCCR5LMNAALDH1A1GAA
SCHEMBL4694791 0.82 MAPT (0.47) MAPTCCR5HTTLMNAALDH1A1
SCHEMBL4694816 0.82 CCR5 (0.44) MAPTSMN1; SMN2CCR5HTTL3MBTL1
SCHEMBL4693310 0.82 CCR5 (0.42) MAPTSMN1; SMN2CCR5HTTL3MBTL1
SCHEMBL4695514 0.81 MAPT (0.40) MAPTSMN1; SMN2CCR5HTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed