SCHEMBL4693113

SCHEMBL4693113

CC(C)C(=O)NOc1cc(C(F)(F)F)ncn1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.40
CHKA P35790 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.37
ACACB O00763 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
ATM Q13315 1/20 0.35
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
CNR1 P21554 1/20 0.33
PIK3CA P42336 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
BRAF P15056 1/20 0.32
KDR P35968 1/20 0.32
MAPK14 Q16539 1/20 0.32
TNNI3K Q59H18 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693115 0.73 CA2 (0.39) CA2CHKAACACBNPSR1ALOX5AP
SCHEMBL24637811 0.72 CA2 (0.46) CA2CHKAACACBNPSR1KDM4E
SCHEMBL4693118 0.71 CA2 (0.42) CA2CHKAACACBALOX5APFEN1
SCHEMBL3374778 0.69 PPARD (0.40) CA2CHKACNR1MAPTKMT2A
SCHEMBL23361197 0.68 PKM (0.50) CA2CHKASMN1; SMN2ALDH1A1KMT2A
SCHEMBL15500846 0.66 NOTUM (0.45) CA2CHKASMN1; SMN2KDM4EALDH1A1
SCHEMBL28853431 0.66 LMNA (0.60) CA2SMN1; SMN2NPSR1KDM4EALDH1A1
SCHEMBL30636498 0.66 LMNA (0.60) CA2SMN1; SMN2NPSR1KDM4EALDH1A1
SCHEMBL28788509 0.66 KDM4E (0.45) SMN1; SMN2NPSR1KDM4EALDH1A1HPGD
SCHEMBL29113156 0.65 LMNA (0.43) CA2ALDH1A1MAPTKMT2ABRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed