SCHEMBL4693258

SCHEMBL4693258

NC(=O)Oc1ccccc1C(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 11/20 0.41
HCRTR2 O43614 11/20 0.41
KCNK3 O14649 2/20 0.38
KCNK9 Q9NPC2 2/20 0.38
GAA P10253 2/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.36
CCR5 P51681 1/20 0.36
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695464 0.88 HCRTR1 (0.44) HCRTR1HCRTR2KCNK3KCNK9CCR5
SCHEMBL4691895 0.88 HCRTR1 (0.33) HCRTR1HCRTR2CCR5
SCHEMBL4694116 0.86 HCRTR2 (0.38) HCRTR1HCRTR2CCR5
SCHEMBL4695826 0.85 HCRTR1 (0.47) HCRTR1HCRTR2KMT2A
SCHEMBL4690142 0.83 MAPK14 (0.41) HCRTR1HCRTR2MAPK14
SCHEMBL4690995 0.83 LMNA (0.38) HCRTR1HCRTR2POLBKMT2ALMNA
SCHEMBL4692504 0.82 HCRTR1 (0.44) HCRTR1HCRTR2GAAKMT2ALMNA
SCHEMBL4690347 0.82 HCRTR2 (0.42) HCRTR1HCRTR2CCR5
SCHEMBL4693757 0.82 LMNA (0.39) HCRTR1HCRTR2LMNACCR5
SCHEMBL4694094 0.81 CHRNB2 (0.44) GAACCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed