SCHEMBL4690995

SCHEMBL4690995

NC(=O)Nc1ccccc1C(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
CCR5 P51681 4/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 4/20 0.35
KDM4E B2RXH2 1/20 0.35
HCRTR1 O43613 2/20 0.35
HCRTR2 O43614 2/20 0.35
RBP4 P02753 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KMT2A Q03164 2/20 0.35
NPC1 O15118 1/20 0.35
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694116 0.86 HCRTR2 (0.38) CCR5HCRTR1HCRTR2CHRNB2CHRNB4
SCHEMBL4694255 0.85 NAMPT (0.43) CCR5MAPTKMT2AMEN1CHRNB2
SCHEMBL4693258 0.83 HCRTR1 (0.41) LMNACCR5HCRTR1HCRTR2CYP2C9
SCHEMBL4693757 0.82 LMNA (0.39) LMNACCR5HCRTR1HCRTR2RBP4
SCHEMBL4690347 0.82 HCRTR2 (0.42) CCR5HCRTR1HCRTR2
SCHEMBL4694094 0.81 CHRNB2 (0.44) CCR5SMN1; SMN2L3MBTL1CHRNB2CHRNB4
SCHEMBL4695377 0.80 CCR5 (0.37) CCR5CYP2C9CYP2C19TSHRCHRNB2
SCHEMBL4691741 0.80 HCRTR2 (0.36) CCR5HCRTR1HCRTR2
SCHEMBL4692504 0.80 HCRTR1 (0.44) LMNACCR5KDM4EHCRTR1HCRTR2
SCHEMBL4694315 0.80 HCRTR2 (0.41) HCRTR1HCRTR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed