SCHEMBL4693311

SCHEMBL4693311

NC(=O)C1[C@@H]2CN(C(=O)c3cccs3)CC2CN1CC[CH]c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
RAB9A P51151 1/20 0.40
HTT P42858 1/20 0.38
CCR5 P51681 1/20 0.38
KCNA5 P22460 1/20 0.37
GAA P10253 1/20 0.37
KDM4E B2RXH2 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5232784 0.87 CHRNB2 (0.43) ALDH1A1SMN1; SMN2
SCHEMBL4692752 0.85 HTT (0.39) ALDH1A1SMN1; SMN2NPC1MAPTRAB9A
SCHEMBL4691561 0.84 CHRM2 (0.36) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL5233804 0.83 DPP4 (0.43) L3MBTL1
SCHEMBL4691769 0.83 CYP2C9 (0.41) CCR5CYP2C9CYP2C19
SCHEMBL4692004 0.82 CHRNB2 (0.34) RAB9ACYP2D6
SCHEMBL5235903 0.82 CCR5 (0.40) SMN1; SMN2NPC1CCR5KDM4EHSD17B10
SCHEMBL5231921 0.82 P2RX7 (0.40) ALDH1A1RAB9AHTTCCR5KCNA5
SCHEMBL5233193 0.81 HTT (0.42) ALDH1A1MAPTHTTCYP2D6CYP2C9
SCHEMBL5235949 0.81 KMT2A (0.34) ALDH1A1SMN1; SMN2CCR5KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed