SCHEMBL4693540

SCHEMBL4693540

COc1cc(F)c(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.37
TNF P01375 3/20 0.35
HCRTR1 O43613 4/20 0.35
HCRTR2 O43614 4/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
CPS1 P31327 7/20 0.34
MCHR1 Q99705 1/20 0.33
MGLL Q99685 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692329 0.92 CCR5 (0.44) CCR5TNFHCRTR1HCRTR2MEN1
SCHEMBL4694815 0.91 HCRTR1 (0.37) CCR5TNFHCRTR1HCRTR2MAPT
SCHEMBL4690309 0.90 HCRTR1 (0.38) CCR5TNFHCRTR1HCRTR2MEN1
SCHEMBL4694788 0.89 HCRTR1 (0.45) CCR5TNFHCRTR1HCRTR2MAPT
SCHEMBL4689519 0.86 ALDH1A1 (0.47) TNFHCRTR1HCRTR2MEN1ALDH1A1
SCHEMBL4694763 0.86 HCRTR1 (0.37) CCR5TNFHCRTR1HCRTR2MAPT
SCHEMBL4693896 0.86 HCRTR1 (0.47) CCR5TNFHCRTR1HCRTR2MEN1
SCHEMBL4690927 0.85 HCRTR1 (0.49) HCRTR1HCRTR2MEN1ALDH1A1LMNA
SCHEMBL3281863 0.84 HCRTR1 (0.48) CCR5TNFHCRTR1HCRTR2
SCHEMBL4690403 0.84 HCRTR1 (0.39) CCR5TNFHCRTR1HCRTR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed