SCHEMBL4690309

SCHEMBL4690309

COc1cc(OC)c(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)c(OC)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 7/20 0.38
HCRTR2 O43614 7/20 0.38
CCR5 P51681 1/20 0.37
PDE4A P27815 3/20 0.37
PDE4B Q07343 3/20 0.37
PDE4C Q08493 3/20 0.37
PDE4D Q08499 3/20 0.37
TNF P01375 3/20 0.37
RORC P51449 5/20 0.37
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692329 0.93 CCR5 (0.44) HCRTR1HCRTR2CCR5PDE4APDE4B
SCHEMBL4693896 0.92 HCRTR1 (0.47) HCRTR1HCRTR2CCR5PDE4APDE4B
SCHEMBL4693540 0.90 CCR5 (0.37) HCRTR1HCRTR2CCR5TNFMEN1
SCHEMBL4695901 0.90 HCRTR2 (0.47) HCRTR1HCRTR2
SCHEMBL4691836 0.88 HCRTR2 (0.40) HCRTR1HCRTR2PDE4APDE4BPDE4C
SCHEMBL4689519 0.87 ALDH1A1 (0.47) HCRTR1HCRTR2TNFMEN1ALDH1A1
SCHEMBL4690927 0.86 HCRTR1 (0.49) HCRTR1HCRTR2MEN1ALDH1A1LMNA
SCHEMBL4691405 0.86 HCRTR1 (0.48) HCRTR1HCRTR2PDE4APDE4BPDE4C
SCHEMBL4694334 0.85 HCRTR1 (0.43) HCRTR1HCRTR2CCR5TNF
SCHEMBL3281863 0.85 HCRTR1 (0.48) HCRTR1HCRTR2CCR5TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed