SCHEMBL4694020

SCHEMBL4694020

CC1CN(Cc2ccc(C(=O)N(C)CCOC(=O)N(c3ccccc3-c3ccccc3)N3CC[CH]CC3)cc2)CC(C)O1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.40
KDM4E B2RXH2 2/20 0.40
POLB P06746 2/20 0.40
HTT P42858 1/20 0.40
BLM P54132 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ACHE P22303 3/20 0.38
AGTR1 P30556 1/20 0.38
AGTR2 P50052 1/20 0.38
MLNR O43193 3/20 0.37
CYP3A4 P08684 2/20 0.37
BCHE P06276 3/20 0.36
MCHR1 Q99705 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280124 0.88 CHRM2 (0.46) CHRM2ACHEBCHEMCHR1
SCHEMBL4692594 0.87 CHRM2 (0.42) CHRM2KDM4EPOLBALDH1A1ACHE
SCHEMBL6021912 0.85 CHRM2 (0.56) CHRM2KDM4EALDH1A1ACHEBCHE
SCHEMBL4693819 0.85 CHRM2 (0.42) CHRM2ALDH1A1ACHEBCHEMCHR1
SCHEMBL4694973 0.84 MCHR1 (0.40) CHRM2POLBACHEBCHEMCHR1
SCHEMBL4692420 0.83 MCHR1 (0.38) CHRM2KDM4EPOLBALDH1A1ACHE
SCHEMBL4695275 0.81 CHRM2 (0.35) CHRM2KDM4EALDH1A1MCHR1
SCHEMBL6021990 0.81 CHRM2 (0.41) CHRM2
SCHEMBL5273742 0.78 NAMPT (0.35) CHRM2KDM4E
SCHEMBL2639275 0.75 CHRM2 (0.45) CHRM2KDM4EALDH1A1ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893577-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2008-03-05 EP claimed
WO-2006138218-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-12-28 WO claimed
EP-1893577-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2008-03-05 EP disclosed
WO-2006138218-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-12-28 WO disclosed