SCHEMBL4694237

SCHEMBL4694237

N[C@@H](CCN1CC2CN(C(=O)C3CC(=O)N(Cc4ccccc4)C3)CC2C1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
ALDH1A1 P00352 3/20 0.44
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HTT P42858 2/20 0.43
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
GLA P06280 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690190 0.88 POLB (0.49) ALDH1A1PKMHTT
SCHEMBL4692279 0.85 CCR5 (0.44) NPC1
Cyclopentane SCHEMBL4695376 0.85 CCR5 (0.52) OPRM1OPRD1SMN1; SMN2
SCHEMBL5231957 0.82 CCR5 (0.65)
SCHEMBL4693061 0.81 CCR5 (0.51) ALDH1A1
SCHEMBL4692082 0.80 CCR5 (0.54)
SCHEMBL4693210 0.80 CCR5 (0.56)
SCHEMBL4691540 0.79 CCR5 (0.56) ALDH1A1
SCHEMBL4690448 0.78 GRIN2B (0.41) ALDH1A1
SCHEMBL3282848 0.78 GRIN2B (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed