SCHEMBL4690448

SCHEMBL4690448

N[C@@H](CCN1CC2CN(C(=O)C3CN(Cc4ccccc4)CCO3)CC2C1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.41
DRD4 P21917 5/20 0.41
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
AGTR2 P50052 1/20 0.39
GRN P28799 1/20 0.39
SORT1 Q99523 1/20 0.39
CYP2C19 P33261 1/20 0.38
MOGAT2 Q3SYC2 1/20 0.38
TACR1 P25103 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
CCR2 P41597 1/20 0.38
KCNH2 Q12809 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CCR5 P51681 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689612 0.83 PKM (0.49) KDM4EALDH1A1HPGDCCR5
SCHEMBL5233175 0.82 CCR5 (0.63) CCR5
SCHEMBL4690443 0.79 GRIN2B (0.37) GRIN2BDRD4DRD2DRD3GRN
SCHEMBL4694237 0.78 OPRM1 (0.47) ALDH1A1
SCHEMBL4694987 0.78 GRIN2B (0.51) GRIN2BDRD2DRD3TACR1CYP2D6
SCHEMBL3282848 0.78 GRIN2B (0.51) GRIN2BDRD2DRD3TACR1CYP2D6
SCHEMBL13779975 0.77 TSHR (0.50) GRIN2BDRD4DRD2DRD3CYP2C19
SCHEMBL4693061 0.77 CCR5 (0.51) ALDH1A1CYP2D6CCR5
SCHEMBL13176328 0.77 CYP2C19 (0.51) GRIN2BDRD4DRD2DRD3CYP2C19
SCHEMBL4690721 0.76 CCR5 (0.45) ALDH1A1HPGDCCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed