SCHEMBL4690190

SCHEMBL4690190

CC(C)CN1CC(C(=O)N2CC3CN(CC[C@H](N)c4ccccc4)CC3C2)CC1=O

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.49
ALDH1A1 P00352 1/20 0.41
CCR5 P51681 7/20 0.41
CCL5 P13501 2/20 0.41
CYP1A2 P05177 1/20 0.41
MAPK1 P28482 1/20 0.41
P2RX7 Q99572 2/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694237 0.88 OPRM1 (0.47) ALDH1A1HTTPKM
SCHEMBL4692279 0.88 CCR5 (0.44) CCR5CCL5MAPK1KMT2A
SCHEMBL4693061 0.81 CCR5 (0.51) ALDH1A1CCR5CCL5KMT2A
SCHEMBL4693210 0.80 CCR5 (0.56) CCR5CCL5
SCHEMBL4692082 0.80 CCR5 (0.54) CCR5CCL5KMT2A
SCHEMBL4692063 0.79 CCL5 (0.51) CCR5CCL5
SCHEMBL4691540 0.79 CCR5 (0.56) ALDH1A1CCR5CCL5
SCHEMBL4692852 0.77 CCR5 (0.53) ALDH1A1CCR5CCL5KMT2A
SCHEMBL4692783 0.77 CCR5 (0.60) CCR5CCL5KMT2A
SCHEMBL4690185 0.76 POLB (0.40) POLBALDH1A1CCR5CCL5CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed