SCHEMBL4694388

SCHEMBL4694388

COc1ccc(C(=O)N2CC3CN(CCCNc4ccc(C)c(Cl)c4)CC3C2)c(OC)n1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.43
HPGD P15428 2/20 0.43
TSHR P16473 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HSD17B10 Q99714 2/20 0.43
HCRTR1 O43613 12/20 0.41
HCRTR2 O43614 12/20 0.41
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
NPC1 O15118 1/20 0.39
KCNK3 O14649 1/20 0.38
KCNK9 Q9NPC2 1/20 0.38
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693245 0.88 MAPT (0.39) RAB9ASMN1; SMN2HCRTR1HCRTR2ALDH1A1
SCHEMBL4693141 0.87 ALDH1A1 (0.45) SMN1; SMN2HCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4694383 0.87 SMN1; SMN2 (0.50) RAB9AHPGDTSHRSMN1; SMN2HSD17B10
SCHEMBL4690931 0.85 MAPT (0.51) RAB9ATSHRSMN1; SMN2HCRTR1HCRTR2
SCHEMBL4695902 0.84 HCRTR2 (0.48) HCRTR1HCRTR2ALDH1A1MAPTHTT
SCHEMBL4690506 0.84 HCRTR1 (0.52) TSHRHCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4691406 0.83 HCRTR1 (0.48) TSHRHCRTR1HCRTR2ALDH1A1MAPT
SCHEMBL4691305 0.83 MAPT (0.42) RAB9ASMN1; SMN2HSD17B10HCRTR1HCRTR2
SCHEMBL4690742 0.82 HCRTR1 (0.46) RAB9AHPGDSMN1; SMN2HCRTR1HCRTR2
SCHEMBL4690670 0.82 UBE2M (0.44) RAB9ASMN1; SMN2HCRTR1HCRTR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed