SCHEMBL4691406

SCHEMBL4691406

COc1ccccc1C(=O)N1CC2CN(CCCNc3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.48
HCRTR2 O43614 4/20 0.48
POLB P06746 3/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NPY2R P49146 2/20 0.45
ALDH1A1 P00352 3/20 0.45
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
CHRM5 P08912 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 2/20 0.41
TACR2 P21452 1/20 0.41
NPC1 O15118 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693956 0.93 HCRTR1 (0.49) HCRTR1HCRTR2POLBMEN1KMT2A
SCHEMBL4692628 0.92 HCRTR1 (0.50) HCRTR1HCRTR2POLBALDH1A1GAA
SCHEMBL4694353 0.91 KCNK3 (0.46) HCRTR1HCRTR2KMT2AALDH1A1KCNK3
SCHEMBL4692337 0.91 HCRTR1 (0.51) HCRTR1HCRTR2POLBMEN1KMT2A
SCHEMBL4693697 0.91 HCRTR1 (0.51) HCRTR1HCRTR2NPY2RALDH1A1GAA
SCHEMBL4690506 0.90 HCRTR1 (0.52) HCRTR1HCRTR2ALDH1A1KCNK3KCNK9
SCHEMBL4691874 0.90 ALDH1A1 (0.43) HCRTR1HCRTR2ALDH1A1KCNK3KCNK9
SCHEMBL4691840 0.90 MAPT (0.47) HCRTR1HCRTR2POLBALDH1A1GAA
SCHEMBL4695902 0.90 HCRTR2 (0.48) HCRTR1HCRTR2ALDH1A1GAAMAPT
SCHEMBL4693901 0.90 HCRTR1 (0.47) HCRTR1HCRTR2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed