SCHEMBL4694462

SCHEMBL4694462

Cc1onc(-c2ccccc2Cl)c1C(=O)N1CC2CN(CC[C@H](N)c3ccccc3)CC2C1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.60
NPC1 O15118 1/20 0.60
EPAS1 Q99814 1/20 0.55
LMNA P02545 5/20 0.55
HTT P42858 2/20 0.55
USP2 O75604 1/20 0.54
CCR5 P51681 1/20 0.53
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.52
GAA P10253 2/20 0.52
KDM4E B2RXH2 1/20 0.51
TSHR P16473 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
RAB9A P51151 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691646 0.88 LMNA (0.59) ALDH1A1LMNAHTTUSP2CCR5
SCHEMBL4691441 0.85 CCR5 (0.67) ALDH1A1LMNAUSP2CCR5KMT2A
SCHEMBL4691805 0.81 CCR5 (0.65) CCR5
SCHEMBL4690784 0.80 CCR5 (0.68) CCR5
SCHEMBL4696787 0.79 CCR5 (0.53) CCR5
SCHEMBL4692749 0.77 CCR5 (0.55) CCR5
SCHEMBL4689905 0.77 CCR5 (0.52) CCR5KMT2AMEN1RAB9A
SCHEMBL3285413 0.77 CCR5 (0.70) CCR5
SCHEMBL3290682 0.77 CCR5 (0.70) CCR5
SCHEMBL3284143 0.77 CCR5 (0.57) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed