SCHEMBL4694987

SCHEMBL4694987

N[C@@H](CCN1CC2CN(Cc3ccccc3)CC2C1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 3/20 0.51
FUCA1 P04066 2/20 0.46
HRH3 Q9Y5N1 1/20 0.46
CYP2D6 P10635 1/20 0.45
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
TACR1 P25103 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3282848 1.00 GRIN2B (0.51) GRIN2BFUCA1HRH3CYP2D6DRD2
SCHEMBL4694382 0.87 SIGMAR1 (0.52) GRIN2B
SCHEMBL4690451 0.83 CCR5 (0.44) CYP2D6
SCHEMBL13326688 0.83 GRIN2B (0.50) GRIN2B
SCHEMBL3283544 0.81 CYP2D6 (0.45) GRIN2BHRH3CYP2D6
SCHEMBL4690721 0.81 CCR5 (0.45)
SCHEMBL5242542 0.81 FUCA1 (0.64) GRIN2BFUCA1HRH3DRD2DRD3
SCHEMBL4692842 0.81 GBA1 (0.43) CYP2D6
SCHEMBL18462977 0.80 FUCA1 (0.51) GRIN2BFUCA1HRH3DRD2DRD3
SCHEMBL21848108 0.79 FUCA1 (0.50) GRIN2BFUCA1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed