SCHEMBL4695897

SCHEMBL4695897

COCC(=O)NC(CCN1CC2CNC[C@H]2[C@H]1C(=O)c1c(C)cccc1C)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.46
TSHR P16473 1/20 0.39
SSTR4 P31391 1/20 0.35
SLC6A9 P48067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694923 0.90 CCR5 (0.56) CCR5SLC6A9
SCHEMBL4692299 0.87 CCR5 (0.58) CCR5SLC6A9
SCHEMBL4696921 0.79 CCR5 (0.47) CCR5SLC6A9
SCHEMBL4694831 0.77 CCR5 (0.41) CCR5
SCHEMBL4696469 0.77 CCR5 (0.41) CCR5
SCHEMBL4693075 0.75 CCR5 (0.80) CCR5
SCHEMBL4693072 0.75 CCR5 (0.80) CCR5
SCHEMBL4696815 0.74 CCR5 (0.40) CCR5
SCHEMBL4695429 0.74 CCR5 (0.46) CCR5SLC6A9
SCHEMBL4695320 0.73 CCR5 (0.41) CCR5SLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed