SCHEMBL4695947

SCHEMBL4695947

C=CCn1ncc2c1CN(C(=O)O)C/C2=N/OCc1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 2/20 0.33
SIGMAR1 Q99720 2/20 0.33
NAMPT P43490 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ALKBH1 Q13686 1/20 0.31
TEAD3 Q99594 2/20 0.31
GPBAR1 Q8TDU6 1/20 0.31
APOBEC3G Q9HC16 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695949 1.00 TMEM97 (0.33) TMEM97SIGMAR1NAMPTNPC1RAB9A
SCHEMBL4143859 0.90 LMNA (0.35)
SCHEMBL4143855 0.90 LMNA (0.35)
SCHEMBL4697047 0.74 ELANE (0.34)
SCHEMBL4695166 0.74 NPBWR1 (0.36)
SCHEMBL5260871 0.72 CHRM2 (0.31)
SCHEMBL20237058 0.69 NPC1 (0.48) NAMPTNPC1RAB9A
SCHEMBL5254817 0.67 TMEM97 (0.35) TMEM97SIGMAR1
SCHEMBL4142491 0.65 KDM1A (0.38)
SCHEMBL20557593 0.65 NPC1 (0.33) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed