SCHEMBL4696003

SCHEMBL4696003

Clc1cc(CBr)c2ccsc2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
HTR2C P28335 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CHEK1 O14757 2/20 0.33
AURKA O14965 2/20 0.33
DAPK3 O43293 2/20 0.33
JAK2 O60674 2/20 0.33
ABL1 P00519 2/20 0.33
NTRK1 P04629 2/20 0.33
CSF1R P07333 2/20 0.33
RET P07949 2/20 0.33
IGF1R P08069 2/20 0.33
PDGFRB P09619 2/20 0.33
PIM1 P11309 2/20 0.33
FGFR1 P11362 2/20 0.33
PRKACA P17612 2/20 0.33
KDR P35968 2/20 0.33
MAP2K2 P36507 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16685781 0.76 CYP2D6 (0.39) CYP2D6CYP2C19HTR2CCYP1A2CYP2C9
SCHEMBL832390 0.69 MAOA (0.47) CYP2D6CYP2C19CYP1A2IGF1RALDH1A1
SCHEMBL2419272 0.68 POLB (0.44) CYP1A2ALDH1A1KMT2A
SCHEMBL32686267 0.68 HTR2C (0.36) CYP2D6CYP2C19HTR2CCYP1A2CYP2C9
SCHEMBL22446422 0.67 LMNA (0.43) CYP2D6CYP2C19CYP1A2CYP2C9CHEK1
SCHEMBL8141883 0.67 ACHE (0.40) CYP2D6CYP2C19CYP1A2CYP2C9ALK
SCHEMBL11347720 0.67 KDM4E (0.40) CYP2C19CYP2C9LMNAALDH1A1MAPT
SCHEMBL11555797 0.66 CYP2A6 (0.34) ALDH1A1
SCHEMBL31221719 0.66 CAMKK1 (0.38) CYP2D6CYP2C19HTR2CCYP1A2CYP2C9
SCHEMBL29244675 0.66 CYP2D6 (0.37) CYP2D6CYP2C19HTR2CCYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937673-A1 IMIDAZOLE DERIVATIVES AS INHIBITORS OF TAFIA Sanofi-Aventis (FR) 2008-07-02 EP disclosed
WO-2007045339-A1 IMIDAZOLE DERIVATIVES AS INHIBITORS OF TAFIA SANOFI-AVENTIS (DE) 2007-04-26 WO disclosed