SCHEMBL4696167

SCHEMBL4696167

CON(C(=O)O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
CRHBP P24387 3/20 0.53
CRHR2 Q13324 3/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
ATM Q13315 1/20 0.53
TLR9 Q9NR96 1/20 0.53
TDP1 Q9NUW8 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GAA P10253 1/20 0.46
MAPK1 P28482 2/20 0.46
CES1 P23141 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
TSHR P16473 1/20 0.44
PHLPP2 Q6ZVD8 1/20 0.44
CES2 O00748 1/20 0.43
SRD5A2 P31213 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5285266 0.80 ALDH1A1 (0.45) ALDH1A1CRHBPCRHR2L3MBTL1MEN1
SCHEMBL2148173 0.77 ALDH1A1 (0.41) ALDH1A1CRHBPCRHR2L3MBTL1MEN1
SCHEMBL1532324 0.77 ALDH1A1 (0.58) ALDH1A1CRHBPCRHR2L3MBTL1MEN1
SCHEMBL29182467 0.76 ALDH1A1 (0.57) ALDH1A1CRHBPCRHR2L3MBTL1MEN1
SCHEMBL7821980 0.76 ALDH1A1 (0.52) ALDH1A1CRHBPCRHR2L3MBTL1MEN1
Hydrochloric Acid SCHEMBL11844609 0.75 ALDH1A1 (0.56) ALDH1A1CRHBPCRHR2L3MBTL1MEN1
SCHEMBL8977870 0.74 MAPT (0.53) ALDH1A1CRHBPCRHR2L3MBTL1MEN1
SCHEMBL3397567 0.74 ALDH1A1 (0.65) ALDH1A1CRHBPCRHR2L3MBTL1MEN1
SCHEMBL20582642 0.73 CRHBP (0.53) ALDH1A1CRHBPCRHR2TDP1SMN1; SMN2
SCHEMBL29667979 0.73 ALDH1A1 (0.51) ALDH1A1CRHBPCRHR2L3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115260211-B Thiophene condensed ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2024-02-06 CN disclosed
CN-115260211-A Thiophene fused ring containing derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-01 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed
EP-1957487-A1 NOVEL PYRIDOPYRAZINES AND THEIR USE AS MODULATORS OF KINASES AEterna Zentaris GmbH (DE) 2008-08-20 EP disclosed
WO-2007054556-A1 NOVEL PYRIDOPYRAZINES AND THEIR USE AS MODULATORS OF KINASES ÆTERNA ZENTARIS GMBH (DE) 2007-05-18 WO disclosed
EP-1785423-A1 Pyridopyrazine derivatives and their use as kinase modulators Zentaris GmbH (DE) 2007-05-16 EP disclosed