SCHEMBL4696280

SCHEMBL4696280

C=CCONC1CN(C(=O)O)Cc2c1cnn2-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
KMT2A Q03164 3/20 0.39
ALPL P05186 1/20 0.39
ALPI P09923 1/20 0.39
ALPG P10696 1/20 0.39
MEN1 O00255 2/20 0.39
DHODH Q02127 3/20 0.38
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5255401 0.83
SCHEMBL4695506 0.79 NPC1 (0.38) NPC1KMT2AALPLALPIALPG
SCHEMBL4651353 0.79 GAA (0.33) KMT2AMEN1
Hydrochloric Acid SCHEMBL4133551 0.78 NPC1 (0.37) NPC1KMT2AALPLALPIALPG
SCHEMBL5255776 0.77 HSD11B1 (0.32)
SCHEMBL4695519 0.77 TMEM97 (0.33)
SCHEMBL4692428 0.74 KEAP1 (0.44) NPC1KEAP1NFE2L2
SCHEMBL5257162 0.74
SCHEMBL5253467 0.72 ALDH1A1 (0.33)
SCHEMBL5186984 0.71 BCDIN3D (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed