SCHEMBL4696597

SCHEMBL4696597

O=C(O)C1NCC(NOCc2ccccc2)c2ccsc21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
EPHX2 P34913 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HTR2C P28335 1/20 0.32
MC4R P32245 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
NAAA Q02083 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4136748 0.90 TSHR (0.34) NPC1RAB9ASMN1; SMN2HTR2CALDH1A1
SCHEMBL5330841 0.83 TSHR (0.40) NPC1RAB9AEPHX2HTR2CMC4R
SCHEMBL4694770 0.78 NPC1 (0.35) NPC1RAB9AEPHX2HTR2CMC4R
SCHEMBL4695714 0.78 NPC1 (0.33) NPC1RAB9AEPHX2HTR2CMC4R
SCHEMBL4695715 0.78 NPC1 (0.33) NPC1RAB9AEPHX2HTR2CMC4R
SCHEMBL4697074 0.76 NPC1 (0.34) NPC1RAB9AEPHX2SMN1; SMN2ALDH1A1
SCHEMBL5187221 0.75 NPC1 (0.37) NPC1RAB9AEPHX2SMN1; SMN2HTR2C
SCHEMBL4693843 0.73 KEAP1 (0.40) NPC1RAB9AALDH1A1
SCHEMBL5252045 0.73 EPHX2 (0.34) NPC1RAB9AEPHX2SMN1; SMN2HTR2C
SCHEMBL5258725 0.73 EPHX2 (0.34) NPC1RAB9AEPHX2SMN1; SMN2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed
EP-1798231-A2 Intermediate products for the preparation of antibacterial compounds NOVEXEL (FR) 2007-06-20 EP disclosed
EP-1399444-B1 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS NOVEXEL (FR) 2007-04-11 EP disclosed